SCHEMBL19983253

SCHEMBL19983253

COC(C)(C)C(=O)NC(CCCCNC(=O)OC(C)(C)C)C(=O)COc1ccon1

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.49
CTSL P07711 1/20 0.45
TDP1 Q9NUW8 6/20 0.44
ATM Q13315 2/20 0.44
MAPT P10636 3/20 0.41
NPSR1 Q6W5P4 5/20 0.41
POLB P06746 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.40
PAX8 Q06710 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21152672 1.00 CTSK (0.49) CTSKCTSLTDP1ATMMAPT
SCHEMBL22460388 0.97 CTSK (0.47) CTSKCTSLTDP1ATMMAPT
SCHEMBL22460387 0.97 CTSK (0.47) CTSKCTSLTDP1ATMMAPT
SCHEMBL22460570 0.87 CTSK (0.42) CTSKCTSLTDP1ATMMAPT
SCHEMBL19972814 0.85 CTSK (0.66) CTSKCTSL
SCHEMBL19972817 0.85 CTSK (0.66) CTSKCTSL
SCHEMBL22445762 0.85 CTSK (0.49) CTSKCTSL
SCHEMBL22445759 0.85 CTSK (0.49) CTSKCTSL
SCHEMBL19983251 0.84 CTSK (0.47) CTSKCTSLTDP1ATMMEN1
SCHEMBL19983282 0.82 CTSK (0.62) CTSKTDP1ATMPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053353-A1 KETONE INHIBITORS OF LYSINE GINGIPAIN Cortexyme, Inc. (US) 2018-03-22 WO disclosed