SCHEMBL19987222

SCHEMBL19987222

CC(C)OC(=O)[C@H](C)NP(=O)(OC[C@H]1OC2(F)C([C@@H]2n2cnc3c(N)ncnc32)C1(C)CCN)Oc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
BTN3A1 O00481 1/20 0.37
AHCY P23526 1/20 0.35
P2RX3 P56373 4/20 0.35
P2RX4 Q99571 4/20 0.35
P2RX1 P51575 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
STING1 Q86WV6 2/20 0.34
P2RY12 Q9H244 1/20 0.34
FAP Q12884 1/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19987164 0.86 CYP3A4 (0.44) CYP3A4CYP2C9BTN3A1AHCYP2RX3
SCHEMBL19987333 0.84 NT5E (0.45) CYP3A4CYP2C9
SCHEMBL19987319 0.84 CYP3A4 (0.42) CYP3A4CYP2C9BTN3A1P2RX3P2RX2
SCHEMBL21136329 0.81 CYP3A4 (0.48) CYP3A4CYP2C9BTN3A1AHCYP2RY12
SCHEMBL21136331 0.81 CYP3A4 (0.48) CYP3A4CYP2C9BTN3A1AHCYP2RY12
SCHEMBL19987217 0.81 CYP3A4 (0.48) CYP3A4CYP2C9BTN3A1AHCYP2RY12
SCHEMBL19987310 0.81 CYP3A4 (0.48) CYP3A4CYP2C9BTN3A1AHCYP2RX3
SCHEMBL19987288 0.81 CYP3A4 (0.44) CYP3A4CYP2C9BTN3A1AHCYP2RX3
SCHEMBL22224910 0.79 CYP3A4 (0.44) CYP3A4CYP2C9BTN3A1AHCYP2RY12
SCHEMBL21136231 0.79 CYP3A4 (0.44) CYP3A4CYP2C9BTN3A1AHCYP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018049535-A1 NUCLEOSIDE ANALOGUES AND METHODS OF USE THEREOF LCB PHARMA INC. (CA) 2018-03-22 WO disclosed