SCHEMBL19987318

SCHEMBL19987318

COC(=O)c1ccc2c(c1)nc(C)n2Cc1ccc(OC)cc1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.68
DCTPP1 Q9H773 3/20 0.62
MAPT P10636 4/20 0.54
GAA P10253 1/20 0.53
NPC1 O15118 1/20 0.53
NLRP3 Q96P20 1/20 0.53
HDAC1 Q13547 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
PPARG P37231 3/20 0.52
KIF11 P52732 1/20 0.52
TDP1 Q9NUW8 1/20 0.51
BRD4 O60885 1/20 0.50
CNR2 P34972 1/20 0.50
RORC P51449 1/20 0.50
DHFR P00374 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025911 0.89 KDM4E (0.70) KDM4EDCTPP1NPC1HDAC1HDAC6
SCHEMBL2161533 0.88 KDM4E (0.68) KDM4EDCTPP1MAPTGAANPC1
SCHEMBL29343401 0.88 KDM4E (0.61) KDM4EDCTPP1MAPTGAANPC1
SCHEMBL29342743 0.88 KDM4E (0.64) KDM4EDCTPP1MAPTPPARGKIF11
SCHEMBL4532827 0.86 PPARG (0.68) KDM4EDCTPP1MAPTHDAC1HDAC6
SCHEMBL12004096 0.85 KDM4E (0.52) KDM4EDCTPP1MAPTNPC1NLRP3
SCHEMBL8036225 0.83 PPARG (0.65) KDM4EMAPTHDAC1HDAC6PPARG
SCHEMBL6172139 0.82 DCTPP1 (0.60) KDM4EDCTPP1MAPTGAANPC1
SCHEMBL1731129 0.81 KDM4E (1.00) KDM4EMAPTGAANPC1TDP1
SCHEMBL17195873 0.81 CFTR (0.59) KDM4EMAPTPPARGKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018053161-A1 NOVEL SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS D-AMINO ACID OXIDASE (DAAO) INHIBITORS NATIONAL TAIWAN UNIVERSITY (TW) 2018-03-22 WO disclosed