SCHEMBL19992145

SCHEMBL19992145

CN1CCCC2C1CCN2C

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.47
CHRNB4 P30926 3/20 0.41
CHRNA3 P32297 3/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNA7 P36544 1/20 0.41
L3MBTL3 Q96JM7 1/20 0.41
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20939371 1.00 CHRM2 (0.47) CHRM2CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL20384062 0.94 CHRM2 (0.45) CHRM2CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2274269 0.94 CHRM2 (0.45) CHRM2CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL17888212 0.88 ALDH1A1 (0.45) CHRM2CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL2274680 0.87 ALDH1A1 (0.36) CHRM2ALDH1A1L3MBTL1
SCHEMBL3436941 0.85 ALDH1A1 (0.46) CHRM2ALDH1A1L3MBTL1
SCHEMBL24781112 0.83 CHRM2 (0.40) CHRM2CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL16063078 0.82 CYP1A2 (0.46) CHRM2ALDH1A1L3MBTL1
SCHEMBL16063087 0.82 CYP1A2 (0.46) CHRM2ALDH1A1L3MBTL1
SCHEMBL15918974 0.81 ALDH1A1 (0.48) CHRM2L3MBTL3ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3512858-B1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2023-11-08 EP disclosed
US-20230339902-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 C4 THERAPEUTICS, INC. (US) 2023-10-26 US disclosed
US-20230339902-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 C4 THERAPEUTICS, INC. (US) 2023-10-26 US disclosed
EP-4242211-A1 IMIDAZOTHIAZOLE COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF Guangzhou Henovcom Bioscience Co., Ltd. (CN) 2023-09-13 EP disclosed
WO-2022100727-A1 IMIDAZOTHIAZOLE COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 广州市恒诺康医药科技有限公司 2022-05-19 WO disclosed
WO-2021259309-A1 GLP-1 RECEPTOR AGONIST, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 广州市恒诺康医药科技有限公司 2021-12-30 WO disclosed
EP-3805234-A1 AROMATIC HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Guangzhou Henovcom Bioscience Co., Ltd. (CN) 2021-04-14 EP disclosed
US-10975100-B2 Fused bicyclic inhibitors of menin-MLL interaction JANSSEN PHARMACEUTICA NV (BE) 2021-04-13 US disclosed
US-20200172556-A1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2020-06-04 US disclosed
US-10611778-B2 Fused bicyclic inhibitors of menin-MLL interaction JANSSEN PHARMACEUTICA NV (BE) 2020-04-07 US disclosed
US-20190218230-A1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION Janssen Pharmaceultica nv (BE) 2019-07-18 US disclosed
WO-2018050684-A1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2018-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190218230-A1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION MLLT1, BMI1, MEN1 CHRM2 4569/4885CHRNB4 4435/4885CHRNA3 3992/4885
US-10611778-B2 Fused bicyclic inhibitors of menin-MLL interaction MLLT1, BMI1, MEN1 CHRM2 4569/4885CHRNB4 4435/4885CHRNA3 3992/4885
US-20230339902-A1 TRICYCLIC LIGANDS FOR DEGRADATION OF IKZF2 OR IKZF4 IKZF1, IKZF3, IKZF2 CHRM2 4704/4885CHRNB4 3026/4885CHRNA3 3830/4885
US-20200172556-A1 FUSED BICYCLIC INHIBITORS OF MENIN-MLL INTERACTION MLLT1, BMI1, MEN1 CHRM2 4569/4885CHRNB4 4435/4885CHRNA3 3992/4885
US-10975100-B2 Fused bicyclic inhibitors of menin-MLL interaction MLLT1, BMI1, MEN1 CHRM2 4569/4885CHRNB4 4435/4885CHRNA3 3992/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.