SCHEMBL19992155

SCHEMBL19992155

Cc1nc2c(C#N)cc(F)cc2c(=O)[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.49
TYMS P04818 1/20 0.43
KDM4E B2RXH2 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TNKS2 Q9H2K2 6/20 0.38
TNKS O95271 5/20 0.38
GAA P10253 2/20 0.38
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PARP2 Q9UGN5 1/20 0.37
PARP3 Q9Y6F1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19992148 0.82 TNKS (0.35) PARP1KDM4ETNKS2TNKSPARP2
SCHEMBL19992165 0.81 PARP1 (0.57) PARP1TYMSKDM4ECYP1A2CYP2D6
SCHEMBL20404208 0.76 PARP1 (0.64) PARP1TYMSKDM4ECYP1A2CYP2D6
SCHEMBL16310700 0.72 PIK3CD (0.38) CYP1A2CYP2C9CYP2C19
SCHEMBL25112470 0.69 PARP1 (0.54) PARP1TYMSKDM4ECYP1A2CYP2D6
SCHEMBL526063 0.69 PARP1 (0.54) PARP1TYMSKDM4ECYP1A2CYP2D6
SCHEMBL16578756 0.68 FASN (0.36) PARP1KDM4EALDH1A1PARP2PARP3
SCHEMBL4369801 0.67 TYMS (0.72) PARP1TYMSKDM4ETNKS2TNKS
SCHEMBL9514561 0.66 PARP1 (1.00) PARP1TYMSKDM4ECYP1A2CYP2D6
SCHEMBL16309057 0.66 PIK3CD (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3008053-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD CALISTOGA LLC (US) 2018-03-21 EP disclosed