SCHEMBL19992148

SCHEMBL19992148

CPc1nc2c(C#N)cc(F)cc2c(=O)[nH]1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNKS O95271 9/20 0.35
TNKS2 Q9H2K2 9/20 0.35
PARP1 P09874 8/20 0.35
PARP2 Q9UGN5 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
PIK3CD O00329 4/20 0.33
KCNH2 Q12809 2/20 0.32
IP6K1 Q92551 1/20 0.32
IP6K3 Q96PC2 1/20 0.32
IP6K2 Q9UHH9 1/20 0.32
PIK3R1 P27986 1/20 0.32
KDM4E B2RXH2 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
CLK1 P49759 1/20 0.30
CLK2 P49760 1/20 0.30
DYRK1A Q13627 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
DYRK1B Q9Y463 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19992155 0.82 PARP1 (0.49) TNKSTNKS2PARP1PARP2PARP3
SCHEMBL16310700 0.67 PIK3CD (0.38) PIK3CDPIK3R1
SCHEMBL16578756 0.65 FASN (0.36) PARP1PARP2PARP3KDM4E
SCHEMBL16309057 0.63 PIK3CD (0.35) PIK3CDPIK3R1
SCHEMBL19992165 0.62 PARP1 (0.57) TNKSTNKS2PARP1PARP2PARP3
SCHEMBL26017922 0.59 TNKS (0.48) TNKSTNKS2PARP1PARP2PARP3
SCHEMBL20404208 0.58 PARP1 (0.64) TNKSTNKS2PARP1KDM4E
SCHEMBL16858459 0.58 KDM4E (0.44) PARP1KDM4ERXFP1
SCHEMBL30753031 0.57 UPP1 (0.43) TNKSTNKS2PARP1KDM4E
SCHEMBL17570611 0.57 TRPV4 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3008053-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD CALISTOGA LLC (US) 2018-03-21 EP disclosed