SCHEMBL1999523

SCHEMBL1999523

CC(C)(C)NC(=O)OCC(C(=O)Nc1ccc2cnccc2c1)c1ccsc1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.51
ROCK1 Q13464 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3336241 0.87 ROCK2 (0.65) ROCK2ROCK1
SCHEMBL3336238 0.87 ROCK2 (0.65) ROCK2ROCK1
SCHEMBL29192409 0.85 ROCK2 (0.67) ROCK2ROCK1
SCHEMBL1094664 0.83 ROCK2 (0.51) ROCK2ROCK1
SCHEMBL11956270 0.83 ROCK2 (0.58) ROCK2ROCK1
SCHEMBL2775044 0.82 ROCK2 (0.56) ROCK2ROCK1
SCHEMBL1105002 0.81 ROCK2 (0.72) ROCK2ROCK1
SCHEMBL23398166 0.81 ROCK2 (0.47) ROCK2ROCK1
SCHEMBL1096576 0.80 ROCK2 (0.55) ROCK2ROCK1
Hydrochloric Acid SCHEMBL1095012 0.80 ROCK2 (0.71) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326623-A2 BETA-AND GAMMA-AMINO-ISOQUINOLINE AMIDE COMPOUNDS AND SUBSTITUTED BENZAMIDE COMPOUNDS Aerie Pharmaceuticals, Inc. (US) 2011-06-01 EP disclosed
WO-2010011853-A2 BETA-AND GAMMA-AMINO-ISOQUINOLINE AMIDE COMPOUNDS AND SUBSTITUTED BENZAMIDE COMPOUNDS AERIE PHARMACEUTICALS, INC. (US) 2010-01-28 WO disclosed