SCHEMBL19996458

SCHEMBL19996458

Cc1ccc2c(=O)[nH]cc(-c3ccc(NC(=O)N4Cc5ccccc5C4)cc3)c2c1

nearest known ligand 0.80

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.80
NAMPT P43490 10/20 0.69
TAS1R3 Q7RTX0 2/20 0.58
TAS1R1 Q7RTX1 2/20 0.58
TAS1R2 Q8TE23 2/20 0.58
ROCK1 Q13464 6/20 0.56
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3704699 0.89 ROCK2 (1.00) ROCK2NAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL19997298 0.87 ROCK2 (0.86) ROCK2NAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL17321517 0.84 ROCK2 (0.82) ROCK2NAMPTROCK1NPC1RAB9A
SCHEMBL17321515 0.82 ROCK1 (0.80) ROCK2NAMPTROCK1
SCHEMBL17321522 0.82 ROCK1 (0.81) ROCK2NAMPTROCK1
SCHEMBL3709151 0.82 ROCK2 (1.00) ROCK2NAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL6121478 0.81 NAMPT (1.00) ROCK2NAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL3707306 0.81 NAMPT (1.00) ROCK2NAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL3712421 0.79 NAMPT (1.00) ROCK2NAMPTROCK1
SCHEMBL6120719 0.79 NAMPT (1.00) ROCK2NAMPTROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926282-B2 Phthalazinones and isoquinolinones as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-27 US disclosed