SCHEMBL19997142

SCHEMBL19997142

O=Cc1cc(OCCOCCOc2ccnc(C=O)c2)ccn1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
MAPK1 P28482 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
NCF1 P14598 7/20 0.39
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
S1PR4 O95977 2/20 0.34
TSHR P16473 1/20 0.34
ORAI1 Q96D31 1/20 0.33
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2455863 0.83 CYP2D6 (0.45) KDM4EALDH1A1SMN1; SMN2NPC1MAPT
SCHEMBL29956732 0.80 NQO1 (0.41) KDM4EALDH1A1SMN1; SMN2NPC1MAPT
SCHEMBL19282141 0.80 NQO1 (0.41) KDM4EALDH1A1SMN1; SMN2NPC1MAPT
SCHEMBL13097217 0.78 CYP2D6 (0.43) MAPT
SCHEMBL21646059 0.76 ALDH1A1 (0.41) KDM4EMAPK1ALDH1A1SMN1; SMN2MAPT
SCHEMBL21645923 0.76 GSTP1 (0.42) KDM4EALDH1A1TSHR
SCHEMBL1208300 0.76 CCR1 (0.55) KDM4EMAPK1ALDH1A1MAPT
SCHEMBL29601133 0.76 CCR1 (0.55) KDM4EMAPK1ALDH1A1MAPT
SCHEMBL17356164 0.76 CCR1 (0.32) KDM4EALDH1A1SMN1; SMN2
SCHEMBL29992466 0.75 MAOB (0.58) KDM4EMAPK1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926290-B2 Inhibitors of INV(16) leukemia UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2018-03-27 US disclosed