SCHEMBL19997286

SCHEMBL19997286

CCC(=O)c1cnn2cc(OCCN3CCOCC3)ccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.60
GAA P10253 1/20 0.60
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 2/20 0.48
PRKAB2 O43741 5/20 0.47
PRKAG1 P54619 5/20 0.47
PRKAA2 P54646 5/20 0.47
PRKAA1 Q13131 5/20 0.47
PRKAG3 Q9UGI9 5/20 0.47
PRKAG2 Q9UGJ0 5/20 0.47
PRKAB1 Q9Y478 5/20 0.47
THRB P10828 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
KMT2A Q03164 1/20 0.47
THRA P10827 1/20 0.45
PSMB1 P20618 1/20 0.45
PSMB5 P28074 1/20 0.45
FLT1 P17948 3/20 0.45
KDR P35968 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19675120 0.92 GAA (0.53) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL17324797 0.90 KDM4E (0.57) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL21947322 0.90 KDM4E (0.49) SMN1; SMN2GAAALDH1A1KDM4ETHRB
SCHEMBL19902561 0.90 SMN1; SMN2 (0.46) SMN1; SMN2GAAALDH1A1KDM4ETHRB
SCHEMBL19902320 0.89 GAA (0.46) SMN1; SMN2GAAALDH1A1KDM4ETHRB
SCHEMBL15882456 0.88 KDM4E (0.51) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL15882213 0.88 GAA (0.50) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL17321465 0.87 KDM4E (0.50) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL19902686 0.86 SMN1; SMN2 (0.44) SMN1; SMN2GAAALDH1A1KDM4EPRKAB2
SCHEMBL21947319 0.84 SMN1; SMN2 (0.56) SMN1; SMN2GAAALDH1A1KDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926282-B2 Phthalazinones and isoquinolinones as rock inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2018-03-27 US disclosed