SCHEMBL19902686

SCHEMBL19902686

CCC(=O)c1cnn2cc(OCCN3CCOC(C)(C)C3)ccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
ROCK2 O75116 1/20 0.35
PRKAB2 O43741 4/20 0.35
PRKAG1 P54619 4/20 0.35
PRKAA2 P54646 4/20 0.35
PRKAA1 Q13131 4/20 0.35
PRKAG3 Q9UGI9 4/20 0.35
PRKAG2 Q9UGJ0 4/20 0.35
PRKAB1 Q9Y478 4/20 0.35
HRH3 Q9Y5N1 2/20 0.35
TBK1 Q9UHD2 1/20 0.34
GRM2 Q14416 1/20 0.34
DRD3 P35462 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17454471 0.92 KDM4E (0.42) SMN1; SMN2GAAKDM4EALDH1A1ROCK2
SCHEMBL17452713 0.88 KDM4E (0.39) SMN1; SMN2GAAKDM4EALDH1A1ROCK2
SCHEMBL19997286 0.86 SMN1; SMN2 (0.60) SMN1; SMN2GAAKDM4EALDH1A1PRKAB2
SCHEMBL20229638 0.84 THRB (0.35) SMN1; SMN2GAAKDM4EALDH1A1HRH3
SCHEMBL19902336 0.83 GAA (0.38) SMN1; SMN2GAAKDM4EALDH1A1ROCK2
SCHEMBL19902561 0.83 SMN1; SMN2 (0.46) SMN1; SMN2GAAKDM4EALDH1A1HRH3
SCHEMBL21947322 0.83 KDM4E (0.49) SMN1; SMN2GAAKDM4EALDH1A1HRH3
SCHEMBL19902683 0.83 HRH3 (0.42) SMN1; SMN2GAAKDM4EALDH1A1ROCK2
SCHEMBL19902320 0.82 GAA (0.46) SMN1; SMN2GAAKDM4EALDH1A1HRH3
SCHEMBL17324797 0.79 KDM4E (0.57) SMN1; SMN2GAAKDM4EALDH1A1PRKAB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed