SCHEMBL20000652

SCHEMBL20000652

FC(F)(F)c1cc(Oc2ccc(Cl)cc2)ccc1C1(Cn2nc[nH]c2=S)OCCO1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
ESRRA P11474 1/20 0.30
PIK3CA P42336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21113813 0.84 SLC6A2 (0.30) SLC6A4
SCHEMBL20000648 0.77 AR (0.46) ARMAOAMAOBHTR2ASLC6A4
SCHEMBL20031435 0.76 AR (0.38) ARHTR2ASLC6A4KCNH2PIK3CA
SCHEMBL2431530 0.76 CYP3A4 (0.42) HTR2ASLC6A4KCNH2
SCHEMBL21113821 0.75 KDM4E (0.31)
SCHEMBL20000651 0.71 CYP3A4 (0.47) HTR2ASLC6A4KCNH2
SCHEMBL1279615 0.69 CYP3A4 (0.47) HTR2ASLC6A4KCNH2
SCHEMBL1279614 0.69 CYP3A4 (0.53) ARHTR2ASLC6A4KCNH2
SCHEMBL15822641 0.68 CYP3A4 (0.44) ARHTR2ASLC6A4KCNH2
SCHEMBL29741799 0.67 AR (0.50) ARMAOAMAOBHTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018054832-A1 NOVEL TRIAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-03-29 WO disclosed