SCHEMBL20002222

SCHEMBL20002222

CC(OCC1CCNC1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 1/20 0.36
SLC6A1 P30531 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRB2 P47870 2/20 0.35
SLC6A12 P48065 2/20 0.35
SLC6A11 P48066 2/20 0.35
SLC6A13 Q9NSD5 2/20 0.35
GABRA1 P14867 1/20 0.35
GABRR1 P24046 1/20 0.35
GABRA4 P48169 1/20 0.35
CHRM3 P20309 3/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRNA3 P32297 1/20 0.31
CHRNB3 Q05901 1/20 0.31
CHRNA6 Q15825 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16886237 0.83 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL21667896 0.81 SLC6A1 (0.39) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL29159663 0.81 SLC6A1 (0.39) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL21667900 0.81 SLC6A1 (0.39) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL29159673 0.81 SLC6A1 (0.39) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL12395690 0.81 SLC6A1 (0.39) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL20002205 0.78 LIPA (0.32)
SCHEMBL20003641 0.78 SLC6A1 (0.41) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL26010433 0.76 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3SLC6A1GABRA5
SCHEMBL20002206 0.75 CYP1A2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed