SCHEMBL20002387

SCHEMBL20002387

CCCOC(=O)C(Cc1cc(F)cc(F)c1)C(=O)OCC

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.44
MMP8 P22894 1/20 0.41
TDP1 Q9NUW8 4/20 0.38
TSHR P16473 3/20 0.38
MAPK1 P28482 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
ALDH1A1 P00352 4/20 0.38
TP53 P04637 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
NR3C2 P08235 1/20 0.35
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34
NTRK1 P04629 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15261624 0.83 MMP8 (0.42) SMN1; SMN2MMP8TDP1TSHRMAPK1
SCHEMBL15261954 0.78 MMP8 (0.39) MMP8TDP1TSHRMAPK1L3MBTL1
SCHEMBL490688 0.77 CA12 (0.52) SMN1; SMN2MMP8TDP1TSHRMAPK1
SCHEMBL5475645 0.77 MMP8 (0.52) MMP8TDP1TSHRMAPK1L3MBTL1
SCHEMBL2427303 0.76 MEN1 (0.40) SMN1; SMN2MMP8TDP1ALDH1A1TP53
SCHEMBL7436472 0.76 MMP8 (0.54) MMP8TDP1MAPK1ALDH1A1TP53
SCHEMBL2428247 0.75 MDM2 (0.39) SMN1; SMN2MMP8TDP1TSHRMAPK1
SCHEMBL2428438 0.73 CYP3A4 (0.39) MMP8TDP1TSHRMAPK1L3MBTL1
SCHEMBL15262664 0.73 MDM2 (0.38) SMN1; SMN2MMP8TDP1TSHRMAPK1
SCHEMBL1312803 0.73 MMP8 (0.62) SMN1; SMN2MMP8TDP1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018056855-A1 DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2018-03-29 WO disclosed
WO-2018056854-A1 BLOOD-BRAIN BARRIER-PENETRANT DOPAMINE-B-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2018-03-29 WO disclosed