SCHEMBL20002887

SCHEMBL20002887

CC(OCc1ccccc1C(F)(F)F)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.58
MAOB P27338 4/20 0.47
MAOA P21397 1/20 0.47
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
TACR1 P25103 1/20 0.40
POLQ O75417 1/20 0.39
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
ATM Q13315 1/20 0.38
RORC P51449 1/20 0.38
POLB P06746 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
SCN8A Q9UQD0 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18213790 0.85 IDO1 (0.61) IDO1MAOBMAOACARM1PRMT6
SCHEMBL16886247 0.83 IDO1 (0.54) IDO1MAOBMAOACARM1PRMT6
SCHEMBL514613 0.77 IDO1 (0.66) IDO1MAOBMAOACARM1PRMT6
SCHEMBL3088642 0.77 IDO1 (0.70) IDO1MAOBMAOACARM1PRMT6
SCHEMBL20267678 0.76 IDO1 (0.59) IDO1MAOBMAOACARM1PRMT6
SCHEMBL20002888 0.76 NR1I2 (0.41) IDO1RORCSLC6A2SLC6A4SLC6A3
SCHEMBL10202644 0.75 IDO1 (0.58) IDO1MAOBMAOACARM1PRMT6
SCHEMBL23759235 0.74 IDO1 (0.47) IDO1MAOBMAOACARM1PRMT6
SCHEMBL13677273 0.74 IDO1 (0.61) IDO1MAOBMAOACARM1PRMT6
SCHEMBL17986303 0.73 IDO1 (0.66) IDO1MAOBMAOACARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed