SCHEMBL20002888

SCHEMBL20002888

CC(OCc1ccccc1OC(F)(F)F)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
RORC P51449 1/20 0.41
SLC6A3 Q01959 6/20 0.40
SLC6A2 P23975 6/20 0.40
SLC6A4 P31645 5/20 0.40
DRD2 P14416 4/20 0.40
GRIN2B Q13224 2/20 0.38
GRIN1 Q05586 1/20 0.38
VNN1 O95497 1/20 0.38
CYP2D6 P10635 4/20 0.37
KCNH2 Q12809 4/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16886236 0.84 NR1I2 (0.39) NR1I2RORCSLC6A3SLC6A2SLC6A4
SCHEMBL2091982 0.79 IDO1 (0.44) SLC6A3SLC6A2SLC6A4DRD2GRIN2B
SCHEMBL20002887 0.76 IDO1 (0.58) RORCSLC6A3SLC6A2SLC6A4IDO1
SCHEMBL7342115 0.75 GRIN2B (0.41) NR1I2RORCSLC6A3SLC6A2SLC6A4
SCHEMBL1690342 0.75 RIPK1 (0.58) SLC6A3SLC6A2SLC6A4DRD2GRIN2B
SCHEMBL1715651 0.75 IDO1 (0.58) SLC6A3SLC6A2SLC6A4GRIN2BGRIN1
SCHEMBL2091979 0.75 SLC6A3 (0.43) NR1I2RORCSLC6A3SLC6A2SLC6A4
SCHEMBL12356638 0.75 SLC6A2 (0.44) SLC6A3SLC6A2SLC6A4DRD2GRIN2B
SCHEMBL2092982 0.74 GRIN2B (0.43) SLC6A3SLC6A2SLC6A4DRD2GRIN2B
SCHEMBL1046654 0.74 MAPT (0.48) SLC6A3SLC6A2SLC6A4DRD2GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092229-B1 PYRROLIDINYL SULFONE DERIVATIVES AND THEIR USE AS ROR GAMMA MODULATORS BRISTOL MYERS SQUIBB CO (US) 2018-03-28 EP disclosed