SCHEMBL20003368

SCHEMBL20003368

CC1(C)OB(c2ccc(CC(=O)Nc3ccn(Cc4ccc(F)cc4)n3)cc2)OC1(C)C.Nc1ccn(Cc2ccc(F)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 19/20 0.59
CACNA1G O43497 18/20 0.59
CACNA1H O95180 17/20 0.59
NPC1 O15118 1/20 0.48
TP53 P04637 1/20 0.48
RAB9A P51151 1/20 0.48
CACNA1C Q13936 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17316652 0.94 CACNA1I (0.65) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL28127713 0.85 CACNA1G (0.58) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL17316455 0.75 CACNA1I (0.73) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL15416384 0.75 GAA (0.64)
SCHEMBL17316566 0.74 CACNA1I (0.72) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL17316282 0.74 CACNA1I (1.00) CACNA1ICACNA1GCACNA1HCACNA1C
SCHEMBL17316503 0.74 CACNA1H (0.81) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL17316277 0.72 CACNA1I (0.69) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL17316425 0.72 CACNA1I (0.69) CACNA1ICACNA1GCACNA1HNPC1TP53
SCHEMBL17316536 0.72 CACNA1G (0.68) CACNA1ICACNA1GCACNA1HNPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9932314-B2 Pyrazole compounds and their use as T-type calcium channel blockers IDORSIA PHARMACEUTICALS LTD (CH) 2018-04-03 US disclosed