SCHEMBL20003634

SCHEMBL20003634

Cc1cc2nccc(Oc3ccc(NC=O)cc3F)c2cn1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 1/20 0.47
PDGFRA P16234 1/20 0.46
MET P08581 9/20 0.45
AXL P30530 8/20 0.45
KDR P35968 2/20 0.45
ROCK2 O75116 1/20 0.42
FLT3 P36888 1/20 0.42
MERTK Q12866 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19373324 0.86 FGFR2 (0.47) FGFR2PDGFRAMETAXLKDR
SCHEMBL29822421 0.84 FGFR2 (0.67) FGFR2PDGFRAMETAXLKDR
SCHEMBL23617110 0.84 FGFR2 (0.67) FGFR2PDGFRAMETAXLKDR
SCHEMBL10269247 0.82 MET (0.54) FGFR2METAXLKDR
SCHEMBL22521192 0.80 FGFR2 (0.59) FGFR2PDGFRAMETAXLKDR
SCHEMBL23617111 0.78 RET (0.57) FGFR2PDGFRAMETAXLKDR
SCHEMBL22521271 0.76 AXL (0.48) FGFR2PDGFRAMETAXLKDR
SCHEMBL22521159 0.76 MET (0.63) FGFR2METAXLFLT3
SCHEMBL20216782 0.75 MET (0.55) METAXLFLT3
SCHEMBL18516581 0.75 MET (0.64) FGFR2METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299369-A1 PYRIDO-AZAHETERECYDIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2018-03-28 EP disclosed