SCHEMBL20003672

SCHEMBL20003672

Bc1c(N)ccnc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.43
TTK P33981 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
MAPT P10636 2/20 0.37
CASP1 P29466 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
DYRK1A Q13627 2/20 0.34
APLNR P35414 1/20 0.33
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
LOX P28300 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
NCF1 P14598 1/20 0.32
RPS6KA5 O75582 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946870 0.78 AURKA (0.46) AURKATTKAURKBINCENPNOS3
SCHEMBL29424822 0.78 AURKA (0.46) AURKATTKAURKBINCENPNOS3
SCHEMBL25957083 0.77 ALDH1A1 (0.39) MAPTMEN1KMT2AAPLNRCCR1
SCHEMBL30294257 0.77 AURKA (0.44) AURKATTKAURKBINCENPNOS3
Hydrochloric Acid SCHEMBL10850408 0.77 AURKA (0.44) AURKATTKAURKBINCENPNOS3
SCHEMBL7899151 0.77 AURKA (0.44) AURKATTKAURKBINCENPNOS3
SCHEMBL8417801 0.77 AURKA (0.44) AURKATTKAURKBINCENPNOS3
SCHEMBL3380754 0.77 AURKA (0.44) AURKATTKAURKBINCENPNOS3
SCHEMBL2208595 0.75 AURKA (0.43) AURKATTKAURKBINCENPNOS3
SCHEMBL21598414 0.75 AURKA (0.43) AURKATTKAURKBINCENPNOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299369-A1 PYRIDO-AZAHETERECYDIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2018-03-28 EP disclosed