SCHEMBL20004125

SCHEMBL20004125

COc1cc2c(cc1Cl)CC(c1c(C)cccc1C#N)=C(C)C2(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.34
TP53 P04637 1/20 0.33
ALDH1A1 P00352 3/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
EIF2AK1 Q9BQI3 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
PKM P14618 1/20 0.31
SRC P12931 2/20 0.31
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31
KDM4E B2RXH2 2/20 0.30
USP2 O75604 2/20 0.30
CASP3 P42574 1/20 0.30
CASP7 P55210 1/20 0.30
TSHR P16473 1/20 0.30
CLK1 P49759 1/20 0.30
SUV39H2 Q9H5I1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21613408 0.78 AR (0.36) ARALDH1A1GAAMAPT
SCHEMBL897479 0.73 CLK1 (0.35) ALDH1A1GAAMAPTHPGDEIF2AK1
SCHEMBL15061898 0.66 CA1 (0.39) ALDH1A1GAAKDM4E
SCHEMBL28641928 0.66 AR (0.49) ARALDH1A1GAAMAPTPKM
SCHEMBL19608991 0.66 AR (0.49) ARALDH1A1GAAMAPTPKM
SCHEMBL897657 0.65 ALK (0.50)
SCHEMBL7811608 0.64 CA1 (0.36) GAAHPGDEIF2AK1SRC
SCHEMBL27376906 0.62 SRC (0.45) ARALDH1A1GAAMAPTHSP90AA1
SCHEMBL21022697 0.61 TSHR (0.65) ARALDH1A1KDM4EUSP2CASP7
SCHEMBL31548017 0.60 ALK (0.43) GAACLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed