SCHEMBL20004201

SCHEMBL20004201

COc1ccc2c(c1N)C(C)(C)c1[nH]c3cc(Br)ccc3c1C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 7/20 0.43
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA4 P22748 3/20 0.37
CA6 P23280 3/20 0.37
GSK3B P49841 3/20 0.36
CHEK1 O14757 1/20 0.35
CCNB2 O95067 2/20 0.35
CDK1 P06493 2/20 0.35
CCNB1 P14635 2/20 0.35
CDK5 Q00535 2/20 0.35
CDK5R1 Q15078 2/20 0.35
CCNB3 Q8WWL7 2/20 0.35
ACHE P22303 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
TUBB4A P04350 2/20 0.34
TUBB P07437 2/20 0.34
TUBA3C P0DPH7 2/20 0.34
TUBA1B P68363 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16775627 0.89 ALK (0.43) ALKCA1CA2CA4CA6
SCHEMBL20004200 0.85 ALK (0.42) ALKCA1CA2CA4CA6
SCHEMBL7807733 0.85 ALK (0.42) ALKCA1CA2CA4CA6
SCHEMBL1755783 0.85 ALK (0.41) ALKCA1CA2CA4CA6
SCHEMBL897634 0.84 ALK (0.42) ALKCA1CA2CA4CA6
SCHEMBL897744 0.81 ALK (0.50) ALKCA1CA2CA4CA6
SCHEMBL16775676 0.80 ALK (0.47) ALKCA1CA2CA4CA6
SCHEMBL27087539 0.79 ALK (0.48) ALKCA1CA2CA4CA6
SCHEMBL896972 0.78 CDK4 (0.46) ALKCA1CA2CA4CA6
SCHEMBL27087566 0.77 ALK (0.47) ALKCA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed