SCHEMBL20004232

SCHEMBL20004232

CCN(CC)CCOc1cc2c(cc1SN1CCOCC1)C(=O)c1c([nH]c3cc(C#N)ccc13)C2(C)C

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 20/20 0.69
KDR P35968 2/20 0.53
GAK O14976 1/20 0.53
ACOX3 O15254 1/20 0.53
NR1I2 O75469 1/20 0.53
ABCB11 O95342 1/20 0.53
EGFR P00533 1/20 0.53
ESR1 P03372 1/20 0.53
PGR P06401 1/20 0.53
RET P07949 1/20 0.53
ROS1 P08922 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
PHKG2 P15735 1/20 0.53
FER P16591 1/20 0.53
EPHA1 P21709 1/20 0.53
DRD1 P21728 1/20 0.53
SLC6A2 P23975 1/20 0.53
PDE4A P27815 1/20 0.53
SLC6A4 P31645 1/20 0.53
DRD3 P35462 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20366347 0.88 ALK (0.54) ALKKDRGAKACOX3NR1I2
SCHEMBL897383 0.86 ALK (0.72) ALKKDRGAKACOX3NR1I2
SCHEMBL20366524 0.85 ALK (0.74) ALKSRPK2SRPK1EML4
SCHEMBL10272635 0.85 ALK (0.67) ALKKDRGAKACOX3NR1I2
SCHEMBL20004594 0.84 ALK (0.74) ALKKDRGAKACOX3NR1I2
SCHEMBL20004641 0.82 ALK (0.65) ALKKDRGAKACOX3NR1I2
SCHEMBL29962690 0.82 ALK (1.00) ALKKDRGAKACOX3NR1I2
SCHEMBL898582 0.82 ALK (1.00) ALKKDRGAKACOX3NR1I2
SCHEMBL20004159 0.81 ALK (0.58) ALKKDRGAKACOX3NR1I2
SCHEMBL896952 0.80 ALK (0.68) ALKSRPK2SRPK1EML4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed