SCHEMBL20004295

SCHEMBL20004295

COc1ccc2c(c1)C(C)(C)c1[nH]c3ccc(N)cc3c1C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA4 P22748 2/20 0.46
CA6 P23280 2/20 0.46
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.41
GFER P55789 1/20 0.41
KMT2A Q03164 1/20 0.41
GSK3B P49841 6/20 0.41
CCNB2 O95067 5/20 0.41
CDK1 P06493 5/20 0.41
CCNB1 P14635 5/20 0.41
CCNB3 Q8WWL7 5/20 0.41
CDK5 Q00535 5/20 0.41
CDK5R1 Q15078 5/20 0.41
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17066405 0.86 CA1 (0.44) CA1CA2CA4CA6MAPT
SCHEMBL1755953 0.82 CA1 (0.39) CA1CA2CA4CA6MAPT
SCHEMBL20366624 0.82 CA1 (0.41) CA1CA2CA4CA6MAPT
SCHEMBL1755993 0.82 CA1 (0.48) CA1CA2CA4CA6MAPT
SCHEMBL898273 0.81 CA1 (0.41) CA1CA2CA4CA6MAPT
SCHEMBL897276 0.81 CTSV (0.57) CA1CA2CA4CA6MAPT
SCHEMBL897959 0.78 CA1 (0.43) CA1CA2CA4CA6MAPT
SCHEMBL896972 0.78 CDK4 (0.46) CA1CA2CA4CA6MAPT
SCHEMBL1755952 0.76 ALK (0.44) CA1CA2CA4CA6MAPT
SCHEMBL897520 0.76 ALK (0.52) CA1CA2CA4CA6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed