SCHEMBL20005999

SCHEMBL20005999

CCO[C@H]1CCCN(C)C(=O)c2c(O)c(=O)c(C(=O)NCc3ccc(F)cc3F)cn2CC1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 8/20 0.56
CYP3A4 P08684 1/20 0.56
TMEM97 Q5BJF2 1/20 0.56
ABCG2 Q9UNQ0 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24521733 0.87 SLC22A2 (0.61) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL30991652 0.85 SLC22A2 (0.63) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL17265186 0.80 SLC22A2 (0.54) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL22482727 0.79 SLC22A2 (0.57) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL10283865 0.79 SLC22A2 (0.60) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL15928664 0.79
SCHEMBL15928579 0.79
Hydrochloric Acid SCHEMBL15914594 0.79
SCHEMBL24799344 0.78 SLC22A2 (0.51) SLC22A2
SCHEMBL82019 0.77 SLC22A2 (0.69) SLC22A2CYP3A4TMEM97ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2940019-B1 SUBSTITUTED SPIROPYRIDO[1,2-a]PYRAZINE DERIVATIVE AND MEDICINAL USE THEREOF AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2018-03-28 EP disclosed