SCHEMBL20006100

SCHEMBL20006100

CC(C)(C)OC(=O)NC1(CN)CC(CCc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
SIGMAR1 Q99720 3/20 0.40
CTSS P25774 3/20 0.39
CTSK P43235 2/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
AKT1 P31749 2/20 0.39
POLB P06746 1/20 0.39
ATM Q13315 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
NPFFR1 Q9GZQ6 1/20 0.37
NPFFR2 Q9Y5X5 1/20 0.37
DPP8 Q6V1X1 1/20 0.37
DPP9 Q86TI2 1/20 0.37
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18506745 0.84 PPARA (0.43) CA12CA1CA7CA14CTSS
SCHEMBL18506647 0.81 EPHX2 (0.41) CA12CA1CA7CA14CTSS
SCHEMBL10073884 0.75 POLB (0.35) CA12CA1CA7CA14SIGMAR1
SCHEMBL5381278 0.73 PPIA (0.49) CA12CA1CA7CA14SIGMAR1
SCHEMBL18506733 0.72 PPARA (0.45) CA12CA1CA7CA14CTSS
SCHEMBL6167707 0.71 CA12 (0.40) CA12CA1CA7CA14SIGMAR1
SCHEMBL19559839 0.71 ADRB2 (0.52) CA12CA1CA7CA14CTSS
SCHEMBL17691231 0.71 EPHX2 (0.42) CA12CA1CA7CA14CTSS
SCHEMBL1752478 0.70 MEN1 (0.37) CA12CA1CA7CA14CTSK
SCHEMBL7372 0.70 AKT1 (0.46) CA12CA1CA7CA14SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2940019-B1 SUBSTITUTED SPIROPYRIDO[1,2-a]PYRAZINE DERIVATIVE AND MEDICINAL USE THEREOF AS HIV INTEGRASE INHIBITOR JAPAN TOBACCO INC (JP) 2018-03-28 EP disclosed