SCHEMBL20008470

SCHEMBL20008470

Cc1ccc(NC(=O)c2ccnc(C(F)(F)F)c2)cc1-c1cc(NCCO)nc(OC[C@@H](C)O)c1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 20/20 0.66
BRAF P15056 6/20 0.61
PDGFRB P09619 1/20 0.60
ARAF P10398 1/20 0.60
DDR1 Q08345 1/20 0.60
DDR2 Q16832 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17523484 0.82 RAF1 (0.84) RAF1BRAFPDGFRBARAFDDR1
SCHEMBL17523483 0.82 RAF1 (0.84) RAF1BRAFPDGFRBARAFDDR1
SCHEMBL20264698 0.80 RAF1 (1.00) RAF1BRAF
SCHEMBL19529492 0.80 RAF1 (1.00) RAF1BRAFPDGFRBARAFDDR1
SCHEMBL20279920 0.79 RAF1 (0.83) RAF1BRAF
SCHEMBL20264662 0.79 RAF1 (1.00) RAF1BRAF
SCHEMBL20008579 0.79 RAF1 (0.60) RAF1BRAFPDGFRBARAFDDR1
SCHEMBL20009424 0.79 RAF1 (0.60) RAF1BRAFPDGFRBARAFDDR1
SCHEMBL20264471 0.79 RAF1 (0.86) RAF1BRAF
SCHEMBL25230508 0.77 RAF1 (0.66) RAF1BRAFPDGFRBARAFDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed