SCHEMBL20008534

SCHEMBL20008534

C=C/C(=C\C=N/CC(C)(C)F)C(=O)Nc1ccc(C)c(-c2cc(OCCC)nc(N3CCCCC3)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRAF P15056 16/20 0.47
RAF1 P04049 14/20 0.47
PDGFRB P09619 1/20 0.45
ARAF P10398 1/20 0.45
DDR1 Q08345 1/20 0.45
DDR2 Q16832 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21091816 0.73 BRAF (0.64) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL20009429 0.67 KDM4E (0.39) BRAFRAF1
SCHEMBL22487984 0.66 BRAF (0.75) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL25260758 0.66 BRAF (0.72) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL19352092 0.65 BRAF (0.51) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL19352093 0.65 BRAF (0.51) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL22488453 0.64 BRAF (0.75) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL31205504 0.64 BRAF (0.70) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL16100633 0.64 RAF1 (1.00) BRAFRAF1PDGFRBARAFDDR1
SCHEMBL24400749 0.64 BRAF (0.57) BRAFRAF1PDGFRBARAFDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299367-A1 BIARYL AMIDE COMPOUNDS AS KINASE INHIBITORS Novartis AG (CH) 2018-03-28 EP disclosed