SCHEMBL20011218

SCHEMBL20011218

CN1c2ncn(C)c2C(=O)N(CCCc2nc3ccccc3s2)C1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44
DRD2 P14416 11/20 0.43
DRD3 P35462 11/20 0.43
DRD4 P21917 9/20 0.43
HTR1A P08908 6/20 0.43
HTR7 P34969 6/20 0.43
HTR2A P28223 4/20 0.43
HRH1 P35367 3/20 0.43
HTR2B P41595 3/20 0.43
HTR2C P28335 3/20 0.43
ADRA2A P08913 2/20 0.43
ADRA2C P18825 2/20 0.43
SLC6A2 P23975 2/20 0.43
ADRA1A P35348 2/20 0.43
DRD1 P21728 2/20 0.43
ADRA2B P18089 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR1D P28221 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24611645 0.72
SCHEMBL24611659 0.69
SCHEMBL18256023 0.67 HTR2A (0.52) SMN1; SMN2HTR2ALMNACYP1A2
SCHEMBL9641726 0.66 SMN1; SMN2 (0.70) SMN1; SMN2ALOX15HTTDRD2DRD3
SCHEMBL24611657 0.66
SCHEMBL27509034 0.65 SMN1; SMN2 (0.68) SMN1; SMN2ALOX15HTTDRD2DRD3
SCHEMBL24611651 0.65 MEN1 (0.30) SMN1; SMN2
SCHEMBL8422776 0.64 DRD2 (0.57) SMN1; SMN2ALOX15HTTDRD2DRD3
SCHEMBL20358330 0.64 SMN1; SMN2 (0.62) SMN1; SMN2ALOX15HTTDRD2DRD3
SCHEMBL14835424 0.64 SMN1; SMN2 (0.67) SMN1; SMN2ALOX15HTTDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3299371-A1 HYDROXYL PURINE COMPOUNDS AND USE THEREOF GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2018-03-28 EP disclosed