SCHEMBL2002304

SCHEMBL2002304

CC(C)(C)N(C(=O)O)C1CCN(c2ccc(Cl)nc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.45
AKR1C3 P42330 1/20 0.45
CHRNB2 P17787 5/20 0.43
CHRNA4 P43681 5/20 0.43
CHRNB4 P30926 5/20 0.43
CHRNA3 P32297 5/20 0.43
MAPT P10636 1/20 0.40
NOTUM Q6P988 2/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18128887 0.85 GCK (0.42) NOTUMMCHR1
SCHEMBL5090920 0.84 CHRNB2 (0.43) CHRM4AKR1C3CHRNB2CHRNA4CHRNB4
SCHEMBL5096829 0.84 CHRNB2 (0.43) CHRM4AKR1C3CHRNB2CHRNA4CHRNB4
SCHEMBL5096831 0.84 CHRNB2 (0.43) CHRM4AKR1C3CHRNB2CHRNA4CHRNB4
SCHEMBL5090914 0.84 CHRNB2 (0.43) CHRM4AKR1C3CHRNB2CHRNA4CHRNB4
SCHEMBL16399141 0.81 MAPT (0.53) CHRNB2CHRNA4CHRNB4CHRNA3MAPT
SCHEMBL16399143 0.81 MAPT (0.53) CHRNB2CHRNA4CHRNB4CHRNA3MAPT
SCHEMBL3939344 0.81 NPY5R (0.34) NOTUMMCHR1
SCHEMBL16398200 0.80 MCHR1 (0.40) CHRNB2CHRNA4NOTUMMCHR1
SCHEMBL22499863 0.79 HRH3 (0.48) CHRM4NOTUMMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960380-B2 Non-anilinic derivatives of isothiazol-3(2H)-one 1,1-dioxides as liver X receptor modulators ASTRAZENECA AB (SE) 2011-06-14 US disclosed