SCHEMBL20025535

SCHEMBL20025535

CN(C)c1ccc(C#Cc2ccc(C3=CCN(CCC(C)(C(N)=O)S(C)(=O)=O)CC3)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
DRD2 P14416 3/20 0.38
DRD4 P21917 3/20 0.38
DRD3 P35462 3/20 0.38
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
SIGMAR1 Q99720 8/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNA3 P22001 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19989562 0.92 MAPK1 (0.42) MAPK1DRD2DRD4DRD3PPARG
SCHEMBL19989661 0.89 MAPK1 (0.40) MAPK1
SCHEMBL19989583 0.89 MAPK1 (0.40) MAPK1DRD2DRD4DRD3PPARG
SCHEMBL20025216 0.88 MAPK1 (0.46) MAPK1DRD2DRD4DRD3PPARG
SCHEMBL23735030 0.83 DRD2 (0.45) DRD2DRD4DRD3PPARGPPARA
SCHEMBL23735068 0.81 DRD2 (0.43) DRD2DRD4DRD3PPARGPPARA
SCHEMBL19989629 0.81 MEN1 (0.35) MAPK1DRD2DRD4DRD3PPARG
SCHEMBL23734851 0.81 DRD2 (0.45) DRD2DRD4DRD3PPARGPPARA
SCHEMBL20025239 0.80 DRD2 (0.38) DRD2DRD4DRD3PPARGPPARA
SCHEMBL20025573 0.79 MAPK1 (0.47) MAPK1DRD2DRD4DRD3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018062924-A1 TETRAHYDROPYRIDINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS DONG-A ST CO., LTD. (KR) 2018-04-05 WO disclosed