SCHEMBL20031008

SCHEMBL20031008

Cc1cc2nc(-c3ccc4c(c3)c(N3CC5(CN(C)C5)C3)nn4C)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.35
PTGDR2 Q9Y5Y4 8/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
PDE5A O76074 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE1C Q14123 1/20 0.33
PDE3A Q14432 1/20 0.33
CYP1A2 P05177 3/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2C19 P33261 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
PMP22 Q01453 2/20 0.33
HIF1A Q16665 2/20 0.33
RGS12 O14924 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20031016 0.93 KDM4E (0.34) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL17547135 0.91 KDM4E (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL20031010 0.87 KMT2A (0.33) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906008 0.87 TACR1 (0.36) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL20030481 0.87 PTGDR2 (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL20030473 0.86 PTGDR2 (0.35) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19905960 0.85 KDM4E (0.42) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL19906245 0.85 HDAC3 (0.37) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL20030465 0.84 PTGDR2 (0.33) KDM4EPTGDR2ALDH1A1MEN1KMT2A
SCHEMBL20030721 0.84 PTGDR2 (0.32) KDM4EPTGDR2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064080-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING HIV INFECTION GILEAD SCIENCES, INC. (US) 2018-04-05 WO disclosed