SCHEMBL20030465

SCHEMBL20030465

Cc1cc2nc(-c3ccc4c(c3)c(N3CCN(C)CC3=O)nn4C)sc2c(-c2ccc(Cl)cc2)c1CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 6/20 0.33
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
PDE5A O76074 1/20 0.32
PDE1A P54750 1/20 0.32
PDE1B Q01064 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE7A Q13946 1/20 0.32
PDE1C Q14123 1/20 0.32
PDE3A Q14432 1/20 0.32
MCHR1 Q99705 1/20 0.31
AKR1B1 P15121 1/20 0.30
EIF4EBP1 Q13541 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20030950 0.92 KDM4E (0.34) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL17547135 0.89 KDM4E (0.35) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20030473 0.87 PTGDR2 (0.35) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20031008 0.84 KDM4E (0.35) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL19905855 0.84 KDM4E (0.39) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20030463 0.84 CYP3A4 (0.36)
SCHEMBL22506256 0.84 CYP3A4 (0.36)
SCHEMBL19905960 0.84 KDM4E (0.42) PTGDR2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20030918 0.83 KDM4E (0.39) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL20030913 0.83 MCHR1 (0.33) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064080-A1 BENZOTHIAZOL-6-YL ACETIC ACID DERIVATIVES AND THEIR USE FOR TREATING HIV INFECTION GILEAD SCIENCES, INC. (US) 2018-04-05 WO disclosed