SCHEMBL20034423

SCHEMBL20034423

CCOc1ccccc1CC(=O)Nc1nnc(CCCCc2nnc(NC(=O)Cc3ccccc3OC)s2)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GLS O94925 15/20 1.00
CFTR P13569 2/20 0.71
MEN1 O00255 2/20 0.63
POLB P06746 2/20 0.63
CYP2C19 P33261 2/20 0.63
KMT2A Q03164 2/20 0.63
GUSB P08236 1/20 0.63
NPSR1 Q6W5P4 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14987201 0.96 GLS (1.00) GLSCFTR
SCHEMBL15042456 0.94 GLS (1.00) GLSCFTRMEN1POLBCYP2C19
SCHEMBL17193304 0.92 GLS (0.91) GLSCFTRMEN1POLBCYP2C19
SCHEMBL14987152 0.86 GLS (1.00) GLSCFTR
SCHEMBL15043814 0.84 GLS (1.00) GLSCFTRMEN1POLBCYP2C19
SCHEMBL15042328 0.84 GLS (1.00) GLS
SCHEMBL19061853 0.83 CFTR (1.00) GLSCFTRMEN1POLBKMT2A
SCHEMBL16887460 0.81 GLS (0.79) GLS
SCHEMBL15042380 0.81 GLS (1.00) GLSCFTRMEN1POLBCYP2C19
SCHEMBL14987489 0.80 GLS (1.00) GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938267-B2 Heterocyclic inhibitors of glutaminase CALITHERA BIOSCIENCES, INC. (US) 2018-04-10 US disclosed