SCHEMBL20034580

SCHEMBL20034580

C=C(CCSCC)SC(=C)NC(=O)CC(C)C

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLS O94925 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19920290 0.82
SCHEMBL20327872 0.70 ALDH1A1 (0.43) TSHRHPGDSMN1; SMN2ALDH1A1GLS
SCHEMBL19920323 0.69
SCHEMBL16312929 0.68 TSHR (0.43) TSHRHPGDALDH1A1
SCHEMBL5691924 0.64 ALDH1A1 (0.50) NPC1HPGDRAB9ASMN1; SMN2ALDH1A1
SCHEMBL16123443 0.64 CYP2D6 (0.43) TSHRHPGDSMN1; SMN2
SCHEMBL21972899 0.63 MEN1 (0.52) TSHRHPGDSMN1; SMN2ALDH1A1
SCHEMBL16590582 0.61 SMN1; SMN2 (0.42) NPC1HPGDRAB9ASMN1; SMN2ALDH1A1
SCHEMBL15355916 0.60
SCHEMBL18469801 0.60 TSHR (0.37) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9938267-B2 Heterocyclic inhibitors of glutaminase CALITHERA BIOSCIENCES, INC. (US) 2018-04-10 US disclosed