SCHEMBL20034585

SCHEMBL20034585

Cc1ccc(Nc2c(NS(=O)(=O)C3CC3)cc3ocnc3c2F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 5/20 0.39
HRH1 P35367 1/20 0.39
BRAF P15056 5/20 0.38
KIT P10721 1/20 0.35
BRD4 O60885 2/20 0.32
PIK3C3 Q8NEB9 1/20 0.32
TSPO P30536 1/20 0.32
CSF1R P07333 1/20 0.32
CKS1B P61024 2/20 0.32
SKP2 Q13309 2/20 0.32
CTPS1 P17812 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15129697 0.88 IDO1 (0.37) BRAFKIT
SCHEMBL19366938 0.81 CSF1R (0.32) CSF1R
SCHEMBL15129483 0.81 BRAF (0.35) MRGPRX1BRAFKITBRD4CKS1B
SCHEMBL20034598 0.80 MRGPRX1 (0.39) MRGPRX1HRH1BRAFKITCTPS1
SCHEMBL391647 0.80 MRGPRX1 (0.44) MRGPRX1HRH1BRAFKITTSPO
SCHEMBL20034519 0.78 MRGPRX1 (0.37) MRGPRX1HRH1BRAFKITPIK3C3
SCHEMBL20034576 0.77 MAP2K1 (0.49)
SCHEMBL19050669 0.76 MRGPRX1 (0.40) MRGPRX1HRH1BRAFBRD4
SCHEMBL12407095 0.75 MRGPRX1 (0.51) MRGPRX1HRH1BRAFKITTSPO
SCHEMBL19050690 0.75 MRGPRX1 (0.41) MRGPRX1HRH1BRAFKITTSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9937158-B2 Benzoheterocyclic compounds and use thereof SHANGHAI KECHOW PHARMA, INC. (CN) 2018-04-10 US disclosed