SCHEMBL20037153

SCHEMBL20037153

Cc1cc2ccccc2n1CC(=O)OCC(=O)Nc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK6 Q92876 2/20 0.68
PRSS1 P07477 1/20 0.68
PRSS2 P07478 1/20 0.68
PRSS3 P35030 1/20 0.68
ALDH1A1 P00352 2/20 0.53
CYP2C19 P33261 2/20 0.53
KMT2A Q03164 4/20 0.50
MEN1 O00255 3/20 0.50
TSHR P16473 2/20 0.50
HTT P42858 1/20 0.50
MAPK1 P28482 1/20 0.50
MAPT P10636 2/20 0.47
RAB9A P51151 2/20 0.47
TP53 P04637 2/20 0.47
KLK7 P49862 1/20 0.46
NPC1 O15118 1/20 0.46
CYP1A2 P05177 1/20 0.46
HSP90AA1 P07900 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037093 0.86 PRSS1 (0.63) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037275 0.85 KLK6 (0.54) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037018 0.85 KLK6 (0.57) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037022 0.82 KLK6 (0.77) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037270 0.81 KLK6 (1.00) KLK6PRSS1PRSS2PRSS3KMT2A
SCHEMBL1779695 0.81 RAB9A (0.68) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL1757508 0.79 KDM4E (0.59) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037004 0.79 PRSS1 (0.51) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037005 0.78 KLK6 (0.89) KLK6PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL20037222 0.78 PRSS1 (0.49) KLK6PRSS1PRSS2PRSS3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed