SCHEMBL20037455

SCHEMBL20037455

Nc1ccc(C2COCCN2)cn1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.48
DRD3 P35462 4/20 0.48
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43
ATR Q13535 1/20 0.39
DRD4 P21917 1/20 0.37
MTOR P42345 9/20 0.36
PIK3R1 P27986 7/20 0.36
PIK3CA P42336 7/20 0.36
RICTOR Q6R327 6/20 0.36
RPTOR Q8N122 6/20 0.36
MAPKAP1 Q9BPZ7 6/20 0.36
MLST8 Q9BVC4 6/20 0.36
ACVR1 Q04771 1/20 0.35
MAP4K1 Q92918 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037654 1.00 DRD2 (0.48) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL3399522 0.83 PRKACA (0.47) PRKACAPRKACGPRKACBATRACVR1
SCHEMBL27392495 0.81 PRKACA (0.38) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL20038364 0.81 PRKACA (0.38) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL27392494 0.81 PRKACA (0.38) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL18291309 0.81 ACVR1 (0.41) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL20038413 0.81 ACVR1 (0.41) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL30920981 0.81 PRKACA (0.38) DRD2DRD3PRKACAPRKACGPRKACB
SCHEMBL24540899 0.78 NOTUM (0.40) PRKACAPRKACGPRKACBATRACVR1
SCHEMBL29761558 0.78 NOTUM (0.40) PRKACAPRKACGPRKACBATRACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed