SCHEMBL20037537

SCHEMBL20037537

Cc1ccc(N2CCN(C(C)C)CCC2=O)cn1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.47
DRD3 P35462 1/20 0.42
KCNH2 Q12809 1/20 0.42
CACNA2D1 P54289 6/20 0.38
SLC6A2 P23975 5/20 0.38
ELANE P08246 1/20 0.38
AKR1C3 P42330 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HDAC4 P56524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20038205 0.87 DRD3 (0.41) HRH3DRD3KCNH2CACNA2D1SLC6A2
SCHEMBL18291315 0.86 DRD3 (0.41) HRH3DRD3KCNH2CACNA2D1SLC6A2
SCHEMBL20038203 0.85 HRH3 (0.44) HRH3DRD3KCNH2CACNA2D1SLC6A2
SCHEMBL20249339 0.83 HRH3 (0.43) HRH3CACNA2D1SLC6A2AKR1C3KDM4E
SCHEMBL20037546 0.80 DRD3 (0.45) DRD3KCNH2ELANEMAPT
SCHEMBL1727049 0.79 AKR1C3 (0.52) HRH3DRD3KCNH2AKR1C3KDM4E
SCHEMBL20038238 0.78 DRD3 (0.43) HRH3DRD3KCNH2ELANEAKR1C3
SCHEMBL255160 0.78 AKR1C3 (0.51) HRH3DRD3KCNH2ELANEAKR1C3
SCHEMBL15492562 0.77 KDM4E (0.54) HRH3KCNH2KDM4EALDH1A1MAPT
SCHEMBL8356124 0.77 AKR1C3 (0.50) HRH3DRD3KCNH2ELANEAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed