SCHEMBL20037547

SCHEMBL20037547

Cc1ccc(N2CCN(CC(C)(C)O)CCC2=O)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 1/20 0.43
KCNH2 Q12809 1/20 0.43
ACVR1 Q04771 1/20 0.37
ELANE P08246 1/20 0.36
PIK3CA P42336 2/20 0.36
MTOR P42345 2/20 0.36
P2RX7 Q99572 4/20 0.35
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CDK2 P24941 1/20 0.34
AKR1C3 P42330 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
WNT1 P04628 3/20 0.32
GSK3B P49841 3/20 0.32
DYRK1A Q13627 3/20 0.32
CHRM4 P08173 1/20 0.32
GRM4 Q14833 1/20 0.32
TLR9 Q9NR96 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291187 0.89 DRD3 (0.46) DRD3KCNH2ACVR1ELANEPIK3CA
SCHEMBL20038204 0.87 PIK3CA (0.34) DRD3KCNH2ACVR1PIK3CAMTOR
SCHEMBL20249341 0.87 HTT (0.35) DRD3KCNH2ACVR1PIK3CAMTOR
SCHEMBL20038327 0.82 DRD3 (0.47) DRD3KCNH2ELANEPIK3CAMTOR
SCHEMBL20038238 0.81 DRD3 (0.43) DRD3KCNH2ELANEP2RX7AKR1C3
SCHEMBL14930379 0.80 ACVR1 (0.47) ACVR1ELANEPIK3CAMTORCDK4
SCHEMBL20037546 0.80 DRD3 (0.45) DRD3KCNH2ELANEKMT2A
SCHEMBL18291670 0.79 DRD3 (0.48) DRD3KCNH2ELANEP2RX7CHRM4
SCHEMBL20038197 0.76 AR (0.36) DRD3KCNH2ACVR1PIK3CAMTOR
SCHEMBL20249326 0.76 AR (0.36) DRD3KCNH2ACVR1PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed