SCHEMBL20037640

SCHEMBL20037640

Nc1ccc(O[C@@H]2CCCNC2)cn1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.59
CHRNA4 P43681 3/20 0.59
ROCK1 Q13464 6/20 0.56
ROCK2 O75116 2/20 0.56
KCNH2 Q12809 1/20 0.56
ALOX5AP P20292 3/20 0.46
FEN1 P39748 3/20 0.46
PRKX P51817 1/20 0.45
PRKCE Q02156 1/20 0.45
PRKCD Q05655 1/20 0.45
PRKD1 Q15139 1/20 0.45
PRKCZ Q05513 1/20 0.44
CHEK2 O96017 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18291534 0.91 CHRNB2 (0.57) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL20037652 0.91 CHRNB2 (0.57) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL2589101 0.86 SLC6A2 (0.47) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL31508102 0.82 PARP10 (0.46) ALOX5APFEN1
SCHEMBL4018813 0.82 MCHR1 (0.43)
SCHEMBL10255943 0.82 PARP10 (0.46) ALOX5APFEN1
SCHEMBL20037651 0.82 CHRNB2 (0.63) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL20255259 0.82 CHRNB2 (0.59) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL20038172 0.82 CHRNB2 (0.59) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL19041965 0.81 ROCK1 (0.52) CHRNB2CHRNA4ROCK1ROCK2ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3305785-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Teijin Pharma Limited (JP) 2018-04-11 EP disclosed