SCHEMBL2004060

SCHEMBL2004060

CC(C)(C)N(C(=O)O)C1CSc2ccccc2N(Cc2ccccc2)C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.48
GAA P10253 3/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
STAT6 P42226 1/20 0.42
GSK3B P49841 2/20 0.41
ACE P12821 4/20 0.41
MME P08473 3/20 0.41
KMT2A Q03164 2/20 0.41
MITF O75030 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 3/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004057 1.00 XIAP (0.48) XIAPGAAALDH1A1CYP1A2CYP3A4
SCHEMBL1996572 0.90 XIAP (0.44) XIAPGAAALDH1A1GSK3BACE
SCHEMBL1996571 0.90 XIAP (0.44) XIAPGAAALDH1A1GSK3BACE
SCHEMBL1999442 0.83 RIPK1 (0.42) XIAPALDH1A1ACEMMEKMT2A
SCHEMBL1999440 0.83 RIPK1 (0.42) XIAPALDH1A1ACEMMEKMT2A
SCHEMBL12569074 0.74 XIAP (0.57) XIAPACEMMEKMT2A
SCHEMBL3149798 0.74 GSK3B (0.50) XIAPALDH1A1GSK3BACEMME
SCHEMBL3156873 0.74 XIAP (0.62) XIAPGSK3BACEMME
SCHEMBL3156878 0.74 XIAP (0.62) XIAPGSK3BACEMME
SCHEMBL15564775 0.72 XIAP (0.64) XIAPCYP3A4ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960373-B2 2-alkoxy-3,4,5-trihydroxyalkylamide-benzothiazepines preparation thereof, compositions containing them and use thereof SANOFI-AVENTIS (FR) 2011-06-14 US disclosed