SCHEMBL20040944

SCHEMBL20040944

Cc1cc(N2CC(C)OC2=O)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
IDH1 O75874 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
GRM2 Q14416 6/20 0.37
FFAR4 Q5NUL3 1/20 0.37
NOTUM Q6P988 1/20 0.37
RECQL P46063 1/20 0.34
THRB P10828 1/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15542604 0.86 NR2E1 (0.41) BRAFKDRIDH1MAOAGRM2
SCHEMBL15541319 0.85 BRAF (0.40) BRAFKDRIDH1GRM2NOTUM
SCHEMBL15542193 0.75 GRM2 (0.39) BRAFKDRIDH1GRM2
SCHEMBL10104299 0.74 KDM4E (0.46) BRAFKDRFFAR4
SCHEMBL7434269 0.74 MAOA (0.66) MAOAMAOBGRM2
SCHEMBL14540825 0.72 GRM2 (0.55) MAOAMAOBGRM2
SCHEMBL25745795 0.71 FFAR4 (0.45) IDH1FFAR4
SCHEMBL5223171 0.71 MAOA (0.40) IDH1MAOAMAOBGRM2
SCHEMBL9805017 0.70 MAOA (0.43) BRAFKDRMAOAGRM2FFAR4
SCHEMBL9846421 0.70 MAOA (0.54) MAOAMAOBGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2864289-B1 CYCLOPROPANECARBOXAMIDO-SUBSTITUTED AROMATIC COMPOUNDS AS ANTI-TUMOR AGENTS CB THERAPEUTICS INC (KY) 2018-04-11 EP disclosed