SCHEMBL20041830

SCHEMBL20041830

C=C(Cc1cn2ccccc2n1)Nc1ccc(-n2nc(C3CC3)cc2C2CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRACR2A Q9BSW2 10/20 0.54
ORAI1 Q96D31 5/20 0.47
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KCNJ6 P48051 2/20 0.38
KCNJ3 P48549 2/20 0.38
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KCNJ5 P48544 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1897432 0.89 CRACR2A (0.68) CRACR2AORAI1KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL1889277 0.88 CRACR2A (0.67) CRACR2AORAI1KDM4EALDH1A1HPGD
SCHEMBL12661319 0.79 CRACR2A (0.54) CRACR2AORAI1KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL1668853 0.79 CRACR2A (0.55) CRACR2AORAI1ALDH1A1SMN1; SMN2
SCHEMBL12673221 0.77 CRACR2A (0.70) CRACR2AORAI1
Hydrochloric Acid SCHEMBL1668162 0.77 CRACR2A (0.69) CRACR2AORAI1
SCHEMBL20006292 0.71 CRACR2A (0.60) CRACR2AORAI1KCNJ6KCNJ3KCNJ5
SCHEMBL1671387 0.70 CRACR2A (1.00) CRACR2AORAI1KDM4EALDH1A1SMN1; SMN2
SCHEMBL1667970 0.69 CRACR2A (1.00) CRACR2AORAI1
Hydrochloric Acid SCHEMBL1668858 0.69 CRACR2A (0.44) CRACR2AORAI1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509974-B1 PYRAZOLES DERIVATIVES MODULATORS OF CALCIUM RELEASE-ACTIVATED CALCIUM CHANNEL AND METHODS FOR TREATMENT OF NON-SMALL CELL LUNG CANCER RHIZEN PHARMACEUTICALS S A (CH) 2018-04-11 EP disclosed