SCHEMBL20042893

SCHEMBL20042893

Cc1nc(O)c2c(n1)CN(Cc1ccccc1)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.45
CYP3A4 P08684 1/20 0.45
DPP4 P27487 1/20 0.45
C5AR1 P21730 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
MC4R P32245 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX15 P16050 1/20 0.38
CLPP Q16740 2/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13329574 0.88 KMT2A (0.56) C5AR1KMT2AMEN1CYP1A2CLPP
SCHEMBL20042770 0.85 CYP2C19 (0.49) CYP2C19CYP3A4DPP4C5AR1KMT2A
SCHEMBL183674 0.82 CYP2C19 (0.40) CYP2C19CYP3A4DPP4C5AR1KMT2A
SCHEMBL20042772 0.80 CYP2C19 (0.43) CYP2C19CYP3A4DPP4C5AR1KMT2A
SCHEMBL13329647 0.78 KMT2A (0.40) CYP2C19C5AR1KMT2AMEN1LMNA
SCHEMBL5999840 0.76 KMT2A (0.56) C5AR1KMT2AMEN1CLPPGAA
SCHEMBL183618 0.74 P2RX7 (0.53) C5AR1KMT2AMEN1GAAKDM4E
SCHEMBL16260721 0.73 KMT2A (0.59) C5AR1KMT2AMEN1CYP1A2CLPP
SCHEMBL18233741 0.73 KMT2A (0.59) C5AR1KMT2AMEN1CLPPGAA
SCHEMBL19616715 0.73 KMT2A (0.50) C5AR1KMT2AMEN1ALOX15CLPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018066718-A1 THERAPEUTIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-12 WO disclosed