SCHEMBL2004422

SCHEMBL2004422

COc1ccc2c(c1F)c(CC(=O)O)c(C)n2C(=O)C1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 5/20 0.38
AKR1C3 P42330 6/20 0.38
AKR1C2 P52895 6/20 0.38
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
HIF1A Q16665 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.35
AKR1C4 P17516 2/20 0.35
AKR1C1 Q04828 2/20 0.35
MEN1 O00255 2/20 0.35
MAPT P10636 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009837 0.92 AKR1C3 (0.39) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2004524 0.92 AKR1C3 (0.39) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2005335 0.91 AKR1C3 (0.39) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2004542 0.89 AKR1C3 (0.38) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2002989 0.89 PTGDR2 (0.39) PTGIRAKR1C3AKR1C2LMNACYP1A2
SCHEMBL2002715 0.89 AKR1C3 (0.40) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2004436 0.89 PTGS1 (0.40) PTGIRAKR1C3AKR1C2ALDH1A1KDM4E
SCHEMBL2008214 0.86 AKR1C3 (0.35) PTGIRAKR1C3AKR1C2LMNACYP1A2
SCHEMBL2004010 0.82 PTGS1 (0.46) PTGIRAKR1C3AKR1C2KDM4ELMNA
SCHEMBL2001827 0.80 PTGS1 (0.41) AKR1C3AKR1C2ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed