SCHEMBL2002989

SCHEMBL2002989

COc1ccc2c(c1F)c(CC(=O)O)c(C)n2C(=O)C1CCN(C)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 5/20 0.39
PTGIR P43119 4/20 0.38
AKR1C3 P42330 5/20 0.38
AKR1C2 P52895 5/20 0.38
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
HIF1A Q16665 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
AKR1C4 P17516 1/20 0.35
AKR1C1 Q04828 1/20 0.35
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004524 0.91 AKR1C3 (0.39) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2009837 0.91 AKR1C3 (0.39) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2005335 0.90 AKR1C3 (0.39) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2004422 0.89 PTGIR (0.38) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2005041 0.89 PTGS1 (0.40) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2002715 0.88 AKR1C3 (0.40) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2004542 0.88 AKR1C3 (0.38) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2006192 0.87 RIPK1 (0.35) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2005243 0.84 AKR1C3 (0.39) PTGDR2PTGIRAKR1C3AKR1C2LMNA
SCHEMBL2004453 0.82 PTGS1 (0.46) PTGDR2PTGIRAKR1C3AKR1C2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed