SCHEMBL2004598

SCHEMBL2004598

CCOc1ccc2c(c1)c(C(=O)c1noc(-c3cccnc3)n1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 8/20 0.41
ALOX5 P09917 3/20 0.41
S1PR1 P21453 1/20 0.41
NPC1 O15118 3/20 0.40
TP53 P04637 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
PTGES2 Q9H7Z7 1/20 0.39
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPT P10636 3/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002012 0.93 PTGES2 (0.40) ALOX5APALOX5NPC1TP53RAB9A
SCHEMBL2007600 0.92 S1PR1 (0.40) ALOX5APALOX5S1PR1NPC1TP53
SCHEMBL2008218 0.92 ALOX5AP (0.41) ALOX5APALOX5S1PR1CYP3A4CYP2D6
SCHEMBL2007194 0.91 ALOX5AP (0.42) ALOX5APALOX5S1PR1PTGS1PTGS2
SCHEMBL2003533 0.90 S1PR1 (0.44) ALOX5APALOX5S1PR1NPC1TP53
SCHEMBL2004983 0.90 PTGES2 (0.42) ALOX5APALOX5S1PR1NPC1TP53
SCHEMBL2001677 0.89 PTGES2 (0.43) ALOX5APALOX5S1PR1NPC1TP53
SCHEMBL2006720 0.88 ALOX5AP (0.44) ALOX5APALOX5SMN1; SMN2PTGES2CYP3A4
SCHEMBL2005007 0.88 PTGES2 (0.40) ALOX5APALOX5S1PR1PTGES2CYP3A4
SCHEMBL2002524 0.87 S1PR1 (0.43) ALOX5APALOX5S1PR1NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed