SCHEMBL2003533

SCHEMBL2003533

CCOc1ccc2c(c1)c(C(=O)c1noc(-c3cccnc3)n1)c(Cl)n2Cc1ccc(Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.44
NPC1 O15118 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 2/20 0.43
RAB9A P51151 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
ALOX5AP P20292 7/20 0.42
ALOX5 P09917 2/20 0.42
MAPT P10636 5/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
PTGES2 Q9H7Z7 1/20 0.39
CYP19A1 P11511 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005239 0.92 MAPT (0.43) NPC1SMN1; SMN2TP53RAB9ANFKB1
SCHEMBL2004267 0.92 S1PR1 (0.42) S1PR1NPC1SMN1; SMN2TP53RAB9A
SCHEMBL2003154 0.91 ALOX5AP (0.42) S1PR1SMN1; SMN2ALOX5APALOX5MAPT
SCHEMBL2003734 0.91 ALOX5AP (0.42) S1PR1SMN1; SMN2NFKB1ALOX5APALOX5
SCHEMBL2004598 0.90 ALOX5AP (0.41) S1PR1NPC1SMN1; SMN2TP53RAB9A
SCHEMBL2002184 0.90 PTGES2 (0.41) NPC1SMN1; SMN2TP53RAB9AMAPT
SCHEMBL2002164 0.87 ALOX5AP (0.45) ALOX5APALOX5MAPTLMNAPTGES2
SCHEMBL2004059 0.86 S1PR1 (0.46) S1PR1NPC1SMN1; SMN2TP53RAB9A
SCHEMBL2003080 0.86 ALOX5AP (0.41) SMN1; SMN2ALOX5APALOX5MAPTKMT2A
SCHEMBL2004576 0.85 HDAC6 (0.43) NPC1SMN1; SMN2TP53RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed