SCHEMBL2004642

SCHEMBL2004642

NC(=O)C(N)(c1ccccc1)c1nc2ccncc2cc1-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.36
CHUK O15111 3/20 0.36
DHODH Q02127 4/20 0.36
CDK2 P24941 2/20 0.36
CDC7 O00311 2/20 0.36
SLC22A12 Q96S37 1/20 0.36
IKBKE Q14164 1/20 0.36
PKMYT1 Q99640 1/20 0.36
CCNE1 P24864 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
ROCK1 Q13464 2/20 0.35
FGFR1 P11362 2/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
CHEK2 O96017 1/20 0.35
CDK1 P06493 1/20 0.35
CSF1R P07333 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004643 0.74 PARP1 (0.35) DHODHCDK2CDC7CCNE1DBF4
SCHEMBL28156921 0.70 FGFR1 (0.62) IKBKBFGFR1KDRKMT2AHASPIN
SCHEMBL28156867 0.68 TNF (0.44) IKBKBCHUKROCK1FGFR1MAPK1
SCHEMBL8169066 0.66 MAPT (0.58) KMT2A
SCHEMBL20553500 0.65 MAPT (0.41) DHODHSLC22A12KMT2A
SCHEMBL28187425 0.65 TNF (0.41) IKBKBCHUKROCK1FGFR1MAPK1
SCHEMBL1339563 0.65 DHODH (0.52) DHODHCDC7DBF4
SCHEMBL10837807 0.64 FGFR1 (0.49) IKBKBFGFR1CHEK2KMT2ASRC
SCHEMBL5717596 0.64 KDM4E (0.44) IKBKBCHUKCDC7ROCK1FGFR1
SCHEMBL1501769 0.63 AKT1 (0.48) IKBKBDHODHSLC22A12AKT1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075383-A1 INHIBITORS OF AKT ACTIVITY MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed