SCHEMBL2004643

SCHEMBL2004643

NC(=O)C(N)(c1cccc(-c2ccccc2)c1)c1ccc2cnccc2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.35
KIF11 P52732 1/20 0.35
DHODH Q02127 2/20 0.35
CDC7 O00311 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
DBF4 Q9UBU7 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ROCK2 O75116 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN5 P54829 1/20 0.34
MAP2 P11137 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
MAP3K8 P41279 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
KMT2A Q03164 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ASIC3 Q9UHC3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20553500 0.76 MAPT (0.41) DHODHROCK2KDM4CKMT2A
SCHEMBL2004642 0.74 IKBKB (0.36) DHODHCDC7CCNE1CDK2DBF4
SCHEMBL3790263 0.73 KCNN4 (0.41) KIF11ROCK2MAPK10NPC1RAB9A
Hydrochloric Acid SCHEMBL3787410 0.72 KCNN4 (0.39) KIF11ROCK2MAPK10NPC1RAB9A
SCHEMBL13723572 0.68 MKNK1 (0.43) PARP1CDC7CCNE1CDK2DBF4
SCHEMBL13724829 0.68 MKNK1 (0.43) PARP1DHODHALDH1A1SMN1; SMN2PTPN5
SCHEMBL21714414 0.66 IKBKB (0.39) ROCK2KDM4CKMT2A
SCHEMBL10305531 0.66 KCNN4 (0.56) PARP1SMN1; SMN2PTPN1PTPN5
SCHEMBL24394795 0.65 PDE10A (0.40) ALDH1A1MAPK10
SCHEMBL12215972 0.65 RAB9A (0.61) ALDH1A1SMN1; SMN2KMT2AMAPK10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075383-A1 INHIBITORS OF AKT ACTIVITY MERCK SHARP & DOHME CORP. (US) 2011-06-23 WO disclosed